Norgestimate is a rapidly and completely converted prodrug, mainly of norelgestromin (17β-deacetylnorgestimate or levonorgestrel 3-oxime), but also of levonorgestrel (3-keto-17β-deacetylnorgestimate) to a lesser extent (22 ± 6% of an administered dose or about 40–70 μg) [2] and of levonorgestrel acetate (levonorgestrel 17β-acetate) in ...

Norgestimate/ethinyl estradiol (Tri-Mili) is used to prevent pregnancy and to treat acne vulgaris on your skin in women 15 years of age or older who have had their first menstrual period and have...

诺孕酯为白色或类白色结晶粉末，分子式为C23H31NO3 ，密度：1.22g/cm3 ，熔点：216ºC ，沸点：497.9ºC at 760mmHg ，又称诺孕酪，炔诺肟酯。 本品为较新的强效孕激素，与炔雌醇配伍组成避孕药。 作用同炔诺酮，活性比炔诺孕酮稍强。 无雄激素活性，但有抗雌激素作用。 对脂代谢影响小，耐受性良好。 [2] 口服吸收迅速，t1/2约为4h。 [2] 临床用作避孕药效果可靠，周期控制好，不降低HDL，有利于脂质代谢，不增加体重，无雄性症等不良反应。 [2] 有血栓史、心肾肝 …

Ethinyl estradiol and norgestimate combination is used to prevent pregnancy. It is a birth control pill that contains two types of hormones, ethinyl estradiol and norgestimate, and when taken properly, prevents pregnancy.

2025年1月29日 · Ethinyl estradiol and norgestimate is a combination birth control pill containing female hormones that prevent ovulation (the release of an egg from an ovary). ethinyl estradiol and norgestimate also causes changes in your cervical mucus and uterine lining, making it harder for sperm to reach the uterus and harder for a fertilized egg to attach ...

NORGESTIMATE; ETHINYL ESTRADIOL (nor JES ti mate; ETH in il es tra DYE ole) prevents ovulation and pregnancy. It may also be used to treat acne. It belongs to a group of medications called oral contraceptives. It is a combination of the hormones estrogen and progestin.

Take this medication by mouth as directed by your doctor, usually once daily. Pick a time of day that is easy for you to remember, and take your pill at the same time each day. If you are taking the chewable tablet, you may either swallow it whole or chew it thoroughly and swallow.

2021年1月26日 · Norgestimate (NGM) is a testosterone derivative with peculiar receptor activities. This is a narrative review of the available data on the pharmacotherapy of NGM in combined hormonal contraceptives (CHCs) in terms of contraceptive efficacy, venous thromboembolism (VTE) risk, safety, tolerability and bleeding patterns.

Norgestimate is a progestin that suppresses ovulation for contraception and reduces free testosterone to treat moderate acne vulgaris. 7,10,11 The therapeutic index is wide as overdoses are rare. 10,11 Patients should be counselled regarding the risk of vascular problems, liver disease, hypertension, metabolic effects, headaches, and bleeding ...

Norgestimate and ethinyl estradiol tablets 0.18 mg/0.035 mg, 0.215 mg/0.035 mg, 0.25 mg/0.035 mg are indicated for the treatment of moderate acne vulgaris in females at least 15 years of age, who have no known contraindications to oral contraceptive therapy and have achieved menarche.