Propiram (Algeril, Dirame, Bay 4503) [2] is a partial μ-opioid receptor agonist and weak μ antagonist analgesic from the ampromide family of drugs related to other drugs such as phenampromide and diampromide.

Propiram fumarate: 一种Opioid receptors激动剂药物，由Bayer AG (Bayer AG)公司最早进行研发，目前全球最高研发状态为终止，作用机制: Opioid receptors激动剂(阿片样受体激动剂)，治疗领域: 神经系统疾病,皮肤和肌肉骨骼疾病,其他疾病。

Propiram | C16H25N3O | CID 26216 - structure, chemical names, physical and chemical properties, classification, patents, literature, biological activities, safety/hazards/toxicity information, supplier lists, and more.

富马酸异丙吡仑: 一种μ opioid receptor激动剂药物，由Grand Pharmaceutical (China) Co., Ltd. (远大医药（中国）有限公司)公司最早进行研发，目前全球最高研发状态为批准上市，作用机制: μ opioid receptor激动剂 (μ-阿片受体激动剂)，治疗领域: 神经系统疾病,其他疾病，在研适应症: 烧伤,神经痛,术后疼痛，在研机构: 远大医药（中国）有限公司。

Propiram is an orally administered opioid analgesic with partial morphine-like agonist and weak antagonist properties. Analgesic efficacy of propiram, usually 50 or 100mg, appears comparable to that of standard dosages of other oral opioid drugs [i.e. pentazocine, pethidine (meperidine)] in …

Propiram (Algeril) is an opioid analgesic from the ampromide family of drugs. It was invented in the 1970s but was not widely marketed, although it saw some limited clinical use, especially in dentistry. Propiram is an effective analgesic comparable to other drugs such as codeine and pethidine, with a normal dose of around 50-100mg. [1]

Propiram is a non-addictive analgesic for the relief of moderate-to-severe pain. Propiram reached Phase III clinical trials in the United States and Canada, but was discontinued. Propiram is a partial opioid mu receptor agonist.

2012年10月18日 · Available data thus indicate that propiram is an effective, orally administered opioid analgesic suitable for providing relief of acute moderate to severe pain arising from various surgical or gynaecological procedures, and that the drug is likely to become a useful alternative in such conditions where opioid analgesia is appropriate.

(S)-Propiram | C16H25N3O | CID 204541 - structure, chemical names, physical and chemical properties, classification, patents, literature, biological activities, safety/hazards/toxicity information, supplier lists, and more.

Properties: LD50 in mice, rats (mg/kg): 874, 1657 orally (Tettenborn). NOTE: This is a controlled substance (opiate): 21 CFR, 1308.11. Therap-Cat: Analgesic (narcotic). Keywords: Analgesic (Narcotic).